| Published Papers |
| No. | Ｔitle URL, Journal, Vol( No), Start Page- End Page, Publication date, DOI
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| 1 | Hexylsilane-mediated direct amidation of amino acids with a catalytic amount of 1,2,4-triazole. , Organic & biomolecular chemistry, 22( 4), 703- 707, Jan. 24, 2024, https://doi.org/10.1039/d3ob01722b |
| 2 |
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| 3 | Amidation of α-Amino Acids Using Dichloro(methyl)(3,3,3-trifluoropropyl)silane and Imidazole without Conventional Protection and Deprotection of α-Amino Group  , Synlett, 33( 15), 1563- 1569, Sep. 2022, https://doi.org/10.1055/a-1865-1792 |
| 4 | Synthesis and Evaluation of Quinone Derivatives for Activity against <i>Trypanosome cruzi</i> , Chemical and Pharmaceutical Bulletin, 69( 12), 1195- 1199, Dec. 1, 2021, https://doi.org/10.1248/cpb.c21-00732 |
| 5 | Effects of the Cytoplasm and Mitochondrial Specific Hydroxyl Radical Scavengers TA293 and mitoTA293 in Bleomycin-Induced Pulmonary Fibrosis Model Mice , Antioxidants, 10( 9), 1398- 1398, Aug. 31, 2021, https://doi.org/10.3390/antiox10091398 |
| 6 |
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| 7 | Acidic Solvent-free Removal of Amine-protecting Diphenylmethyl Groups in the Presence of Camphorsulfonic Acid , CHEMISTRY LETTERS, 46( 10), 1456- 1458, Oct. 2017, https://doi.org/10.1246/cl.170604 |
| 8 | Asymmetric Synthesis of CP-99,994 by Ring-expanding Amination of Monosubstituted Prolinols , CHEMISTRY LETTERS, 45( 1), 54- 56, Jan. 2016, https://doi.org/10.1246/cl.150940 |
| 9 | Synthesis and biological evaluation of quinones derived from natural product komaroviquinone as anti-Trypanosoma cruzi agents , BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 25( 15), 2967- 2971, Aug. 2015, https://doi.org/10.1016/j.bmcl.2015.05.022 |
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| 11 |
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| 12 |
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| 13 |
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| 14 | Catalytic asymmetric epoxidation of alpha,beta-unsaturated phosphane oxides with a Y(O-iPr)3/biphenyldiol complex , CHEMISTRY-AN ASIAN JOURNAL, 3( 8-9), 1500- 1504, 2008, https://doi.org/10.1002/asia.200800035 |
| 15 | Activation and Utilization of Carbon Dioxide , Bull. Takasaki University of Health and Welfare, 7, 199- 209, 2008, |
| 16 |
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| 17 | Cyclopentyl methyl ether as a new and alternative process solvent , ORGANIC PROCESS RESEARCH & DEVELOPMENT, 11( 2), 251- 258, Mar. 2007, https://doi.org/10.1021/op0680136 |
| 18 | Bismuth-catalyzed direct substitution of the hydroxy group in alcohols with sulfonamides, carbamates, and carboxamides , ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 46( 3), 409- 413, 2007, https://doi.org/10.1002/anie.200602909 |
| 19 | Bismuth- and hafnium-catalyzed hydroamination of vinyl arenes with sulfonamides, carbamates, and carboxamides , CHEMISTRY-AN ASIAN JOURNAL, 2( 1), 150- 154, 2007, https://doi.org/10.1002/asia.200600284 |
| 20 | syn-selective direct catalytic asymmetric Mannich-type reactions of aromatic and heteroaromatic hydroxy ketones promoted by Y[N(SiMe3)(2)](3)/linked-BINOL complexes , BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, 79( 12), 1906- 1912, Dec. 2006, https://doi.org/10.1246/bcsj.79.1906 |
| 21 |
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| 22 | Mixed La-Li heterobimetallic complexes for tertiary nitroaldol resolution , JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 128( 36), 11776- 11777, Sep. 2006, https://doi.org/10.1021/ja064858l |
| 23 | Catalytic asymmetric epoxidation of alpha,beta-unsaturated N-acylpyrroles as monodentate and activated ester equivalent acceptors , TETRAHEDRON, 62( 28), 6630- 6639, Jul. 2006, https://doi.org/10.1016/j.tet.2005.12.074 |
| 24 | Bismuth-catalyzed intermolecular hydroamination of 1,3-dienes with carbamates, sulfonamides, and carboxamides , JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 128( 5), 1611- 1614, Feb. 2006, https://doi.org/10.1021/ja056112d |
| 25 |
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| 26 | Nickel-catalyzed homoallylation of aldehydes with 1,3-dienes: (anti-3-Methyl-1-phenyl-4-penten-1-ol and anti-5-Methyl-1-phenyl-6-hepten-3-ol) , Organic Syntheses, 83, 88- 96, 2006, https://doi.org/10.15227/orgsyn.083.0088 |
| 27 | Bismuth-catalyzed intermolecular hydroamination of 1,3-dienes with carbarnates, sulfonamides, and carboxamides (vol 128, pg 1611, 2006) , Journal of the American Chemical Society, 128( 12), 4162- , 2006, https://doi.org/10.1021/ja060684w |
| 28 | syn-selective direct catalytic asymmetric Mannich-type reactions of hydroxyketones using Y{N(SiMe3)(2)}(3)/linked-BINOL complexes , ORGANIC LETTERS, 7( 23), 5339- 5342, Nov. 2005, https://doi.org/10.1021/ol052384+ |
| 29 | Lewis acid-Lewis acid heterobimetallic cooperative catalysis: Mechanistic studies and application in enantioselective aza-Michael reaction , JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 127( 38), 13419- 13427, Sep. 2005, https://doi.org/10.1021/ja054066b |
| 30 | Catalytic asymmetric cyano-ethoxycarbonylation reaction of aldehydes using a YLi(3)Tris(binaphthoxide) (YLB) complex: Mechanism and roles of achiral additives , JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 127( 10), 3413- 3422, Mar. 2005, https://doi.org/10.1021/ja042887v |
| 31 | Catalytic asymmetric cyano-phosphorylation of aldehydes promoted by heterobimetallic YLi(3)tris(binaphthoxide) (YLB) complex , SYNLETT, ( 13), 2434- 2436, Nov. 2004, https://doi.org/10.1055/s-2004-832821 |
| 32 | Mechanistic studies of a reaction promoted by the [YLi3{triS(binaphthoxide)}] complex: Are three 1,1 '-Bi-2-naphthol units in a rare-earth-alkali-metal heterobimetallic complex necessary? , ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 43( 34), 4493- 4497, 2004, https://doi.org/10.1002/anie.200454202 |
| 33 | Heterobimetallic catalysis in asymmetric 1,4-addition of O-alkylhydroxylamine to enones , JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 125( 52), 16178- 16179, Dec. 2003, https://doi.org/10.1021/ja038688d |
| 34 | Efficient two-step conversion of alpha,beta-unsaturated aldehydes to optically active gamma-oxy-alpha,beta-unsaturated nitriles and its application to the total synthesis of (+)-patulolide C , ORGANIC LETTERS, 5( 17), 3021- 3024, Aug. 2003, https://doi.org/10.1021/ol034944f |
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| 36 |
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| MISC |
| No. | Ｔitle URL, Journal, Vol( No), Start Page- End Page, Publication date
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| 1 | 天然物コマロビキノン及び関連化合物の骨髄腫細胞に対する抗腫瘍活性の評価 , 日本薬学会年会要旨集, 138年会( 2), 189- 189, Mar. 2018
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| 2 | Tofacitinib合成中間体の立体選択的合成法の検討 , 日本薬学会年会要旨集, 138年会( 2), 174- 174, Mar. 2018
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| 3 | 直鎖型アルキルベンゼンスルホン酸のウシ脳カルシニューリン活性に対する影響 , 日本生化学会大会プログラム・講演要旨集, 89回, [2P- 186], Sep. 2016
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| 4 | 直鎖型アルキルベンゼンスルホン酸のプロテインホスファターゼ活性に対する影響 , 日本生化学会大会・日本分子生物学会年会合同大会講演要旨集, 88回・38回, [3P0515]- [3P0515], Dec. 2015
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| 5 | シャーガス病治療薬の開発を志向したキノン誘導体の合成と活性評価 , 日本薬学会年会要旨集, 135年会( 2), 245- 245, Mar. 2015
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| 6 | Characterization of Alkylbenzene Sulfonate Inhibitors of Protein Phosphatase 1α Activity , Kitakanto Med J, 65( 1), 53- 59, 2015
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| 7 | マイトジェン刺激したJurkat T細胞のサイトカイン産生に対するアルキルベンゼンスルホン酸の効果 , 日本生化学会大会プログラム・講演要旨集, 87回, [4P- 181], Oct. 2014
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| 8 | Catalytic Asymmetric Reactions Using N-Acylpyrroles as Activated Monodentate Ester Surrogates , Proceedings of the Symposium on Progress in Organic Reactions and Syntheses, 31( 0), 162- 162, 2005
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| 9 | Catalytic Asymmetric Conjugate Addition of O-Methylhydroxylamine to α, β-Unsaturated Ketones Using YL_3tris(binaphthoxide) (YLB) Complex , 希土類 = Rare earths, 44, 214- 215, May. 13, 2004
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| Conference Activities & Talks |
| No. | Ｔitle, Conference, Publication date, Promoter, Venue
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| 1 | Amidation of unprotected amino acids using hexylsilane, The 142nd Annual Meeting of the Pharmaceutical Society of Japan, Mar. 27, 2022, ,
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| 2 | Investigation of effects on students about English educational methods including pronunciation of technical terms in pharmacy and organic chemistry, The 142nd Annual Meeting of the Pharmaceutical Society of Japan, Mar. 26, 2022, ,
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| 3 | Design and synthesis of novel two-point recognition host compounds containing guanidino group, The 141st Annual Meeting of the Pharmaceutical Society of Japan, Mar. 29, 2021, ,
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| 4 | Amidation of unprotected amino acids using Dichloro(methyl)(3,3,3-trifluoropropyl)silane, The 141st Annual Meeting of the Pharmaceutical Society of Japan, Mar. 27, 2021, ,
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| 5 | Research for the regiocontrolled synthesis of novel oxatomide derivatives containing 3,8-diazabicyclo[3,2,1]octane structure, The 140th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 28, 2020, ,
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| 6 | Regioselective Epoxidation using Hexafluoroacetone trihydrate, The 140th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 28, 2020, ,
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| 7 | Epoxidation using 3,3,3-Trifluoropyruvate Catalysts, The 140th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 28, 2020, ,
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| 8 | Investigation of reaction mechanism and versatility in diphenylmethyl (DPM) group removal reaction using CSA, The 140th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 28, 2020, ,
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| 9 | Inhibitory effects of oxatomide derivatives on human P2X7 receotor, The 140th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 27, 2020, ,
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| 10 | Design and synthesis of novel indole-replaced oxatomide derivatives with P2X7 inhibitory activity, The 140th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 26, 2020, ,
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| 11 | Design and synthesis of novel two-point recognition host compounds and research to the selective recognition of dicarboxylic acids, The 140th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 26, 2020, ,
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| 12 | Classroom observation and feedback in faculty development, The 139th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 21, 2019, ,
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| 13 | Synthesis and biological evaluation of the natural product komaroviquinone and related compounds aiming at a potential therapeutic lead compound for high-risk multiple myeloma, The 138th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 27, 2018, ,
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| 14 | Asymmetric Synthesis of the Key Intermediate for Tofacitinib, The 138th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 27, 2018, ,
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| 15 | Effect of the bovine brain calcineurin activity of linear alkylbenzene sulfonate, The 89th Annual Meeting of JBS, Sep. 26, 2016, ,
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| 16 | Tackling infectious disease : Structural modification of komaroviquinone to develop novel therapeutic agents for Chagas’ Disease, 8th AFMC International Medicinal Chemistry Symposium AIMECS 11, Frontier of Medicinal Science, Nov. 29, 2011, ,
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| 17 | Efficient Synthesis of Komaroviquinone and its Derivatives, The 130th Annual Meeting of the Pharmaceutical Society of Japan, Mar. 28, 2010, ,
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